1-Tosyl-2-trifluoroacetylindole as Promising Partner for Synthesis of Fused Fluorinated Heterocycles
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We prepared 1-tosyl-2-trifluoroacetylindole - a novel example of an electron-deficient indole with an electrophilic C(3) position. This substance was involved in cyclocondensation with a variety of amidines to propose a new general pathway to 8H-[4,5-b]indolopyrimidines with yield 50-80%. CF3-containing 5H-[3,2-d]indolopyrimidines were unknown before this study.
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2011 ◽
Vol 194-196
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pp. 503-506
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Keyword(s):
2018 ◽
Vol 24
(36)
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pp. 9157-9164
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2010 ◽
Vol 23
(3)
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pp. 540-546
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Keyword(s):
2012 ◽
Vol 77
(9)
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pp. C966-C974
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