Synthesis of 9‐O‐Arylated Berberine with a Polystyrene Resin Supported Copper(II) Catalyst

2021 ◽  
Vol 6 (16) ◽  
pp. 4011-4014
Author(s):  
Qi Meng ◽  
Lian Zhang ◽  
Xinhui Zhu ◽  
Qiaoqiao Teng
Keyword(s):  
1985 ◽  
Vol 15 (8) ◽  
pp. 833-837 ◽  
Author(s):  
Takeshi Noma ◽  
Yutaka Kawano ◽  
Naoko Yoshimura ◽  
Tsutomu Abe ◽  
Kenji Inagaki ◽  
...  

Tetrahedron ◽  
2005 ◽  
Vol 61 (32) ◽  
pp. 7789-7795 ◽  
Author(s):  
Mario Gonçalves ◽  
Karine Estieu-Gionnet ◽  
Georges Laïn ◽  
Mireille Bayle ◽  
Natacha Betz ◽  
...  
Keyword(s):  

1992 ◽  
Vol 57 (8) ◽  
pp. 1707-1718
Author(s):  
Wolfgang Voelter ◽  
Gerhard Breipohl ◽  
Chryssa Tzougraki ◽  
Eveline Jungfleisch-Turgut

The solid phase synthesis of an amidated somatostatin analogue based on the principle of differentiated acidolysis is described. The acid labile and smoothly cleavable t-Bumeoc moiety (1% TFA/DCM) is used for temporary Nα-protection of D- and L-amino acids and [4-[[[9H-fluoren-9-yl-methoxycarbonyl]amino](4-methoxyphenyl)methyl]-2-methylphenoxy]acetic acid, attached to an aminomethylated polystyrene resin is used as acid sensitive linker of the solid carrier which releases the peptide in its amide form by treatment with TFA. Its preparation is described in detail.


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