scholarly journals Design, synthesis, and biological evaluation of abiotic, non-lactone modulators of LuxR-type quorum sensing

2011 ◽  
Vol 19 (16) ◽  
pp. 4812-4819 ◽  
Author(s):  
Christine E. McInnis ◽  
Helen E. Blackwell
Keyword(s):  
Quorum Sensing ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

scholarly journals Design, synthesis and biological evaluation of 1,2,3-triazole based 2-aminobenzimidazoles as novel inhibitors of LasR dependent quorum sensing in Pseudomonas aeruginosa

RSC Advances ◽  
2019 ◽  
Vol 9 (50) ◽  
pp. 29273-29292 ◽  
Author(s):  
Singireddi Srinivasarao ◽  
Adinarayana Nandikolla ◽  
Shashidhar Nizalapur ◽  
Tsz Tin Yu ◽  
Sravani Pulya ◽  
...  
Keyword(s):  
Pseudomonas Aeruginosa ◽  
Quorum Sensing ◽  
Cell Line ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Hek 293 ◽  
Line P ◽  
Synthesis And Biological Evaluation ◽  
Hek 293 Cell Line

Out of 40 benzimdazoles, 12 exhibited potent QSI activity against P. aeruginosa6p, most active QSI is docked to LasR and is less toxic against HEK 293 cell line.

Design, synthesis and biological evaluation of novel unsymmetrical azines as quorum sensing inhibitors

RSC Advances ◽  
2015 ◽  
Vol 5 (97) ◽  
pp. 80027-80038 ◽  
Author(s):  
Sumit S. Chourasiya ◽  
Deepika Kathuria ◽  
Shaminder Singh ◽  
Vijay C. Sonawane ◽  
Asit K. Chakraborti ◽  
...  
Keyword(s):  
Quorum Sensing ◽  
Biological Evaluation ◽  
One Pot ◽  
Design Synthesis ◽  
Quorum Sensing Inhibitors ◽  
Synthesis And Biological Evaluation

In this report, novel unsymmetrical azines have been designed and synthesised by using one pot approach. Further, they were evaluated as quorum sensing inhibitors.

Design, Synthesis and Biological Evaluation of Triazole-Containing 2-Phenylindole and Salicylic Acid as Quorum Sensing Inhibitors Against Pseudomonas aeruginosa

2018 ◽  
Vol 3 (32) ◽  
pp. 9170-9180 ◽  
Author(s):  
Singireddi Srinivasarao ◽  
Shashidhar Nizalapur ◽  
Tsz Tin Yu ◽  
Daniel Stanley Wenholz ◽  
Prakruti Trivedi ◽  
...  
Keyword(s):  
Pseudomonas Aeruginosa ◽  
Salicylic Acid ◽  
Quorum Sensing ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Quorum Sensing Inhibitors ◽  
Synthesis And Biological Evaluation

Design, synthesis and biological evaluation of non-natural modulators of quorum sensing in Pseudomonas aeruginosa

2012 ◽  
Vol 10 (30) ◽  
pp. 6032 ◽  
Author(s):  
James T. Hodgkinson ◽  
Warren R. J. D. Galloway ◽  
Megan Wright ◽  
Ioulia K. Mati ◽  
Rebecca L. Nicholson ◽  
...  
Keyword(s):  
Pseudomonas Aeruginosa ◽  
Quorum Sensing ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

Design, Synthesis and Biological Evaluation of Hybrid Molecules Containing Conjugated Styryl Ketone and α-Bromoacryloyl Moieties

2012 ◽  
Vol 9 (2) ◽  
pp. 140-152 ◽  
Author(s):  
Romeo Romagnoli ◽  
Pier Giovanni Baraldi ◽  
Olga Cruz-Lopez ◽  
Maria Kimatrai Salvador ◽  
Delia Preti ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Design Synthesis ◽  
Hybrid Molecules ◽  
Synthesis And Biological Evaluation
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