Essential structure of orexin 1 receptor antagonist YNT-707: Conversion of the 16-cyclopropylmethyl group to the 16-sulfonamide group in D-nor-nalfurafine derivatives

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2022.128550 ◽

2022 ◽

pp. 128550

Author(s):

Koki Katoh ◽

Noriki Kutsumura ◽

Naoshi Yamamoto ◽

Yasuyuki Nagumo ◽

Tsuyoshi Saitoh ◽

...

Keyword(s):

Receptor Antagonist ◽

Sulfonamide Group

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The novel histamine H2 receptor antagonist FRG-8813 prevents delay of wound repair induced by hydrogen peroxide in a rabbit gastric epithelial cell system

Journal of Gastroenterology and Hepatology ◽

10.1046/j.1440-1746.1998.01735.x ◽

1998 ◽

Vol 13 (11-s4) ◽

pp. S209-S213

Author(s):

NOBUHIRO SATO ◽

SUMIO WATANABE ◽

XIAN-EN WANG ◽

TARO OSADA ◽

HIROSHI TANAKA ◽

...

Keyword(s):

Hydrogen Peroxide ◽

Epithelial Cell ◽

Receptor Antagonist ◽

Wound Repair ◽

Cell System ◽

The Novel ◽

H2 Receptor Antagonist ◽

Histamine H2 Receptor ◽

H2 Receptor ◽

Histamine H2 Receptor Antagonist

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Colonic effects of TAK-637: A novel NK, receptor antagonist

Gastroenterology ◽

10.1016/s0016-5085(01)81646-2 ◽

2001 ◽

Vol 120 (5) ◽

pp. A331-A331

Author(s):

K VENKOVA ◽

K TYLER ◽

D SUTKOWSKIMARKMANN

Keyword(s):

Receptor Antagonist ◽

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Interleukin-1 regulates interleukin-1β/interleukin-1 receptor antagonist mRNA expression in human endometrial stromal cells

Journal of the Society for Gynecologic Investigation ◽

10.1016/s1071-5576(97)86393-9 ◽

1998 ◽

Vol 5 (1) ◽

pp. 116A-116A

Author(s):

H HUANG ◽

Y WEN ◽

J KRUSSEL ◽

H WANG ◽

Y SOONG ◽

...

Keyword(s):

Receptor Antagonist ◽

Mrna Expression ◽

Stromal Cells ◽

Interleukin 1 ◽

Interleukin 1Β ◽

Endometrial Stromal Cells ◽

Interleukin 1 Receptor Antagonist

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Continuous brachial plexus blockade in combination with the NMDA receptor antagonist memantine prevents phantom pain in acute traumatic upper limb amputees

Yearbook of Anesthesiology and Pain Management ◽

10.1016/s1073-5437(08)70995-1 ◽

2008 ◽

Vol 2008 ◽

pp. 265-266

Author(s):

S.E. Abram

Keyword(s):

Nmda Receptor ◽

Brachial Plexus ◽

Receptor Antagonist ◽

Nmda Receptor Antagonist ◽

Phantom Pain ◽

Brachial Plexus Blockade

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Abstract #1229: Effects on Glucose Lowering of a Cortisol Receptor Antagonist in Cushing Syndrome

Endocrine Practice ◽

10.1016/s1530-891x(20)42458-9 ◽

2015 ◽

Vol 21 ◽

pp. 289

Author(s):

Amy Lee

Keyword(s):

Receptor Antagonist ◽

Cushing Syndrome ◽

Glucose Lowering

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Effects of rolofylline, a new adenosine A1 receptor antagonist, on symptoms, renal function and outcomes in patients with acute heart failure. Results of the PROTECT pilot study

European Journal of Heart Failure Supplements ◽

10.1016/s1567-4215(08)60149-6 ◽

2008 ◽

Vol 7 ◽

pp. 53-54

Author(s):

C OCONNOR ◽

G COTTER ◽

H DITTRICH ◽

B DAVISONWEATHERLEY ◽

M METRA ◽

...

Keyword(s):

Heart Failure ◽

Renal Function ◽

Pilot Study ◽

Receptor Antagonist ◽

Acute Heart Failure ◽

Adenosine A1 Receptor ◽

Adenosine A1 ◽

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Microinjection of NMDA Receptor Antagonist AP5 to the Telencephalon

PsycEXTRA Dataset ◽

10.1037/e413802005-463 ◽

2001 ◽

Author(s):

Jennifer Bazner ◽

Min Qi ◽

Xiaojuan Xu

Keyword(s):

Nmda Receptor ◽

Receptor Antagonist ◽

Nmda Receptor Antagonist

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Safety Study of Intraarticular Injection of Interleukin 1 Receptor Antagonist in Patients With Painful Knee Osteoarthritis: A Multicenter Study

Yearbook of Medicine ◽

10.1016/s0084-3873(08)70352-3 ◽

2006 ◽

Vol 2006 ◽

pp. 56-57

Author(s):

M.H. Pillinger

Keyword(s):

Knee Osteoarthritis ◽

Receptor Antagonist ◽

Multicenter Study ◽

Interleukin 1 ◽

Intraarticular Injection ◽

Safety Study ◽

Interleukin 1 Receptor Antagonist ◽

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A chemokine receptor antagonist reduces the incidence and severity of collagen induced arthritis in DBA/1 mice

Immunology Letters ◽

10.1016/s0165-2478(97)86999-4 ◽

1997 ◽

Vol 56 (1-3) ◽

pp. 42-43

Author(s):

C Plater-Zyberk

Keyword(s):

Receptor Antagonist ◽

Chemokine Receptor ◽

Collagen Induced Arthritis ◽

Chemokine Receptor Antagonist

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Chronic hemodynamic and antifibrotic effects of a specific angiotensin II receptor antagonist (losartan) in bile duct ligated (BDL) rats and in portal vein ligated (PVL) rats

Journal of Hepatology ◽

10.1016/s0168-8278(01)80311-1 ◽

2001 ◽

Vol 34 (0) ◽

pp. 88

Author(s):

V Croquet

Keyword(s):

Angiotensin Ii ◽

Bile Duct ◽

Portal Vein ◽

Receptor Antagonist ◽

Angiotensin Ii Receptor ◽

Angiotensin Ii Receptor Antagonist

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