Antitumor studies – Part 2: Structure–activity relationship study for flavin analogs including investigations on their in vitro antitumor assay and docking simulation into protein tyrosine kinase

Activity Relationship ◽

Protein Tyrosine ◽

Structure Activity ◽

New horizons in drug discovery of lymphocyte-specific protein tyrosine kinase (Lck) inhibitors: a decade review (2011–2021) focussing on structure–activity relationship (SAR) and docking insights

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756366.2021.1937143 ◽

2021 ◽

Vol 36 (1) ◽

pp. 1574-1602

Author(s):

Ahmed Elkamhawy ◽

Eslam M. H. Ali ◽

Kyeong Lee

Keyword(s):

Drug Discovery ◽

Tyrosine Kinase ◽

Protein Tyrosine Kinase ◽

Specific Protein ◽

Activity Relationship ◽

Protein Tyrosine ◽

New Horizons ◽

Structure Activity

Structure Activity Relationship Study of Emodin Derivatives Based on the Protein-Tyrosine Kinase and Protein Kinase C Inhibitory Activities and Cytotoxicity

Natural Product Letters ◽

10.1080/10575639708041191 ◽

1997 ◽

Vol 10 (3) ◽

pp. 173-180 ◽

Cited By ~ 3

Author(s):

Darrick S. H. L. Kim ◽

Nuphavan M. Koonchanok ◽

Robert L. Geahlen ◽

Curtis L. Ashendel ◽

Ching-Jer Chang

Keyword(s):

Protein Kinase C ◽

Protein Kinase ◽

Tyrosine Kinase ◽

Protein Tyrosine Kinase ◽

Activity Relationship ◽

Kinase C ◽

Structure Activity ◽

Relationship Study ◽

Inhibitory Activities

Quantitative Structure−Activity Relationship of Flavonoid Analogues. 3. Inhibition of p56lck Protein Tyrosine Kinase

Journal of Chemical Information and Computer Sciences ◽

10.1021/ci000001a ◽

2000 ◽

Vol 40 (4) ◽

pp. 994-1001 ◽

Cited By ~ 50

Author(s):

M. Oblak ◽

M. Randic ◽

T. Solmajer

Keyword(s):

Tyrosine Kinase ◽

Protein Tyrosine Kinase ◽

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Protein Tyrosine ◽

Structure Activity ◽

Structure-activity relationship of a novel peptide substrate for p60c-src protein tyrosine kinase

Letters in Peptide Science ◽

10.1007/bf00142241 ◽

1996 ◽

Vol 2 (5) ◽

pp. 289-296 ◽

Cited By ~ 6

Author(s):

Qiang Lou ◽

Jinzi Wu ◽

Sydney E. Salmon ◽

Kit S. Lam

Keyword(s):

Tyrosine Kinase ◽

Protein Tyrosine Kinase ◽

Activity Relationship ◽

Peptide Substrate ◽

Protein Tyrosine ◽

Structure Activity ◽

Structure–Activity Relationship of Halophenols as a New Class of Protein Tyrosine Kinase Inhibitors

International Journal of Molecular Sciences ◽

10.3390/ijms12096104 ◽

2011 ◽

Vol 12 (9) ◽

pp. 6104-6115 ◽

Cited By ~ 4

Author(s):

Xiu E Feng ◽

Wan Yi Zhao ◽

Shu Rong Ban ◽

Cheng Xiao Zhao ◽

Qing Shan Li ◽

...

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Protein Tyrosine Kinase ◽

Kinase Inhibitors ◽

Activity Relationship ◽

Protein Tyrosine ◽

New Class ◽

Structure Activity ◽

ChemInform Abstract: Quantitative Structure-Activity Relationship of Flavonoid Analogues. Part 3. Inhibition of p56lck Protein Tyrosine Kinase.

ChemInform ◽

10.1002/chin.200042239 ◽

2000 ◽

Vol 31 (42) ◽

pp. no-no

Author(s):

M. Oblak ◽

M. Randic ◽

T. Solmajer

Keyword(s):

Tyrosine Kinase ◽

Protein Tyrosine Kinase ◽

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Protein Tyrosine ◽

Structure Activity ◽

Synthesis, structure–activity relationship, and p210bcr-abl protein tyrosine kinase activity of novel AG 957 analogs☆

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2004.12.003 ◽

2005 ◽

Vol 13 (5) ◽

pp. 1749-1761 ◽

Cited By ~ 18

Author(s):

Gurmeet Kaur ◽

Ven L. Narayanan ◽

Prabhakar A. Risbood ◽

Melinda G. Hollingshead ◽

Sherman F. Stinson ◽

...

Keyword(s):

Tyrosine Kinase ◽

Protein Tyrosine Kinase ◽

Kinase Activity ◽

Activity Relationship ◽

Tyrosine Kinase Activity ◽

Protein Tyrosine ◽

Structure Activity ◽

Protein Tyrosine Kinase Activity

Anti-leishmanial and anti-trypanosomal activities of 1,4-dihydropyridines: In vitro evaluation and structure–activity relationship study

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2010.09.015 ◽

2010 ◽

Vol 18 (22) ◽

pp. 8044-8053 ◽

Cited By ~ 35

Author(s):

Juliana Q. Reimão ◽

Marcus T. Scotti ◽

André G. Tempone

Keyword(s):

Activity Relationship ◽

In Vitro Evaluation ◽

Structure Activity ◽

Radiochemical Investigations of99mTc−N3S-X-BBN[7−14]NH2: An in Vitro/in Vivo Structure−Activity Relationship Study Where X = 0-, 3-, 5-, 8-, and 11-Carbon Tethering Moieties

Bioconjugate Chemistry ◽

10.1021/bc020034r ◽

2003 ◽

Vol 14 (1) ◽

pp. 93-102 ◽

Cited By ~ 63

Author(s):

C. Jeffrey Smith ◽

Hariprasad Gali ◽

Gary L. Sieckman ◽

Chris Higginbotham ◽

Wynn A. Volkert ◽

...

Keyword(s):

Activity Relationship ◽

Structure Activity ◽

Synthesis of tyrosol glycosides and their structure–activity relationship study in biochemical assays and in human cells in vitro

Toxicology Letters ◽

10.1016/j.toxlet.2017.07.331 ◽

2017 ◽

Vol 280 ◽

pp. S118

Author(s):

Eva Horvathova ◽

Eliska Galova ◽

Andrea Sevcovicova ◽

Martina Klapakova ◽

Andrej Bohac ◽

...

Keyword(s):

Human Cells ◽

Activity Relationship ◽

Structure Activity ◽

Biochemical Assays ◽