Design, synthesis, and characterization of novel aminoalcohol quinolines with strong in vitro antimalarial activity

2021 ◽  
pp. 113981
Author(s):  
A. Dassonville-Klimpt ◽  
J. Schneider ◽  
C. Damiani ◽  
C. Tisnerat ◽  
A. Cohen ◽  
...  
Keyword(s):  
Antimalarial Activity ◽  
Synthesis And Characterization ◽  
Design Synthesis

Design, synthesis, and characterization of 6β-naltrexol analogs, and their selectivity for in vitro opioid receptor subtypes

2009 ◽  
Vol 19 (10) ◽  
pp. 2811-2814 ◽  
Author(s):  
Andrea L. Pelotte ◽  
Ryan M. Smith ◽  
Mario Ayestas ◽  
Christina M. Dersch ◽  
Edward J. Bilsky ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Synthesis And Characterization ◽  
Receptor Subtypes ◽  
Design Synthesis ◽  
Opioid Receptor Subtypes

scholarly journals Design, Synthesis and Characterization of Novel Arylamides Containing 1,2,4-triazole Nuclei for Possible Antimicrobial Activity

2004 ◽  
Vol 1 (5) ◽  
pp. 228-230 ◽  
Author(s):  
S. R. Dhol ◽  
P. M. Gami ◽  
R. C. Khunt ◽  
A. R. Parikh
Keyword(s):  
Antimicrobial Activity ◽  
Hydrazine Hydrate ◽  
Carbon Disulfide ◽  
Acid Chloride ◽  
Potassium Hydroxide ◽  
Synthesis And Characterization ◽  
Design Synthesis ◽  
Elemental Analyses

Diphenyl aceto hydrazide on reaction with carbon disulfide and potassium hydroxide gave potassiumα,α-diphenyl acetamido dithiocarbamate, which on cyclisation with hydrazine hydrate yielded key intermediate 3-mercapto-4,N-amino-5-benzhydryl-1,2,4-triazoles. The key intermediate on condensation with different acid chloride afforded our titled compounds. The synthesised compounds have been confirmed elemental analyses and further supported by spectral data. All the synthesised compounds have been evaluated for theirin vitroin vitro antimicrobial activity.

Design, synthesis and characterization of new 1,2,3-triazolyl pyrazole derivatives as potential antimicrobial agents via a Vilsmeier–Haack reaction approach

RSC Advances ◽  
2016 ◽  
Vol 6 (64) ◽  
pp. 59375-59388 ◽  
Author(s):  
Manjunatha Bhat ◽  
Nagaraja G. K. ◽  
Reshma Kayarmar ◽  
Peethamber S. K. ◽  
Mohammed Shafeeulla R
Keyword(s):  
Antimicrobial Agents ◽  
Synthesis And Characterization ◽  
Pyrazole Derivatives ◽  
Design Synthesis ◽  
Anti Oxidant ◽  
Anti Fungal

A new series of 1,2,3-triazolyl pyrazole derivatives were synthesisedviaa Vilsmeier–Haack reaction approach and screened for theirin vitroanti-bacterial, anti-fungal and anti-oxidant activities.

scholarly journals 3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties

2015 ◽  
Vol 94 ◽  
pp. 45-55 ◽  
Author(s):  
Céline Meinguet ◽  
Céline Bruyère ◽  
Raphaël Frédérick ◽  
Véronique Mathieu ◽  
Christelle Vancraeynest ◽  
...  
Keyword(s):  
3D Qsar ◽  
Synthesis And Characterization ◽  
Design Synthesis
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