scholarly journals Discovery of a First-in-Class Potent Small Molecule Antagonist against the Adrenomedullin-2 Receptor

2020 ◽  
Vol 3 (4) ◽  
pp. 706-719
Author(s):  
Paris Avgoustou ◽  
Ameera B. A. Jailani ◽  
Jean-Olivier Zirimwabagabo ◽  
Matthew J. Tozer ◽  
Karl R. Gibson ◽  
...  
Keyword(s):  
Small Molecule ◽  
Small Molecule Antagonist

A small molecule antagonist of ghrelin O-acyltransferase (GOAT)

2011 ◽  
Vol 47 (26) ◽  
pp. 7512 ◽  
Author(s):  
Amanda L. Garner ◽  
Kim D. Janda
Keyword(s):  
Small Molecule ◽  
Small Molecule Antagonist

scholarly journals Idalopirdine – a small molecule antagonist of 5-HT6 with therapeutic potential against obesity

2015 ◽  
Vol 30 (6) ◽  
pp. 1487-1494 ◽  
Author(s):  
Magdalena Dudek ◽  
Monika Marcinkowska ◽  
Adam Bucki ◽  
Adrian Olczyk ◽  
Marcin Kołaczkowski
Keyword(s):  
Small Molecule ◽  
Therapeutic Potential ◽  
Small Molecule Antagonist

scholarly journals Identification of a Novel Small Molecule Antagonist of the Ectopic Olfactory Receptor Olfr78/OR51E2

2021 ◽  
Vol 35 (S1) ◽  
Author(s):  
Alexandra Scharr ◽  
Julisia Chau ◽  
Erwin Ni ◽  
Andy Chang
Keyword(s):  
Small Molecule ◽  
Olfactory Receptor ◽  
Small Molecule Antagonist

The novel small-molecule antagonist MMG-11 preferentially inhibits TLR2/1 signaling

2020 ◽  
Vol 171 ◽  
pp. 113687 ◽  
Author(s):  
Maria Grabowski ◽  
Manuela S. Murgueitio ◽  
Marcel Bermudez ◽  
Gerhard Wolber ◽  
Günther Weindl
Keyword(s):  
Small Molecule ◽  
The Novel ◽  
Small Molecule Antagonist

Identification and Characterization of a Small Molecule Antagonist of Human VPAC2 Receptor

2009 ◽  
Vol 77 (1) ◽  
pp. 95-101 ◽  
Author(s):  
Alan Chu ◽  
Jeremy S. Caldwell ◽  
Yu Alice Chen
Keyword(s):  
Small Molecule ◽  
Small Molecule Antagonist ◽  
Identification And Characterization

scholarly journals A Small-Molecule Antagonist of the β-Catenin/TCF4 Interaction Blocks the Self-Renewal of Cancer Stem Cells and Suppresses Tumorigenesis

2015 ◽  
Vol 76 (4) ◽  
pp. 891-901 ◽  
Author(s):  
Liang Fang ◽  
Qionghua Zhu ◽  
Martin Neuenschwander ◽  
Edgar Specker ◽  
Annika Wulf-Goldenberg ◽  
...  
Keyword(s):  
Stem Cells ◽  
Cancer Stem Cells ◽  
Small Molecule ◽  
The Self ◽  
Self Renewal ◽  
Small Molecule Antagonist

scholarly journals A Small Molecule Antagonist Inhibits Thyrotropin Receptor Antibody-Induced Orbital Fibroblast Functions Involved in the Pathogenesis of Graves Ophthalmopathy

2013 ◽  
Vol 98 (5) ◽  
pp. 2153-2159 ◽  
Author(s):  
Adina F. Turcu ◽  
Seema Kumar ◽  
Susanne Neumann ◽  
Michael Coenen ◽  
Seethalakshmi Iyer ◽  
...  
Keyword(s):  
Small Molecule ◽  
Thyrotropin Receptor ◽  
Receptor Antibody ◽  
Small Molecule Antagonist ◽  
Graves Ophthalmopathy ◽  
Thyrotropin Receptor Antibody ◽  
Orbital Fibroblast

Abstract B03: A small-molecule antagonist of CX3CR1 impairs homing and colonization of breast cancer cells in the skeleton

2016 ◽  
Author(s):  
Fei Shen ◽  
Yun Zhang ◽  
Danielle Jernigan ◽  
Jie Yan ◽  
Fernando Garcia ◽  
...  
Keyword(s):  
Breast Cancer ◽  
Cancer Cells ◽  
Small Molecule ◽  
Breast Cancer Cells ◽  
Small Molecule Antagonist

Chimeric protein probes for C5a receptors through fusion of the anaphylatoxin C5a core region with a small-molecule antagonist

2019 ◽  
Vol 62 (10) ◽  
pp. 1371-1378 ◽  
Author(s):  
Chao Zuo ◽  
Wei-Wei Shi ◽  
Xiao-Xu Chen ◽  
Marie Glatz ◽  
Bernd Riedl ◽  
...  
Keyword(s):  
Small Molecule ◽  
Chimeric Protein ◽  
Core Region ◽  
Small Molecule Antagonist ◽  
Anaphylatoxin C5a ◽  
C5a Receptors
Sign in / Sign up

Export Citation Format

Share Document