Effect of gastric pH and of a moderate CYP3A4 inducer on the pharmacokinetics of daridorexant, a dual orexin receptor antagonist

British Journal of Clinical Pharmacology ◽

10.1111/bcp.15029 ◽

2021 ◽

Author(s):

Martine Gehin ◽

Jolanta Wierdak ◽

Giancarlo Sabattini ◽

Patricia N. Sidharta ◽

Jasper Dingemanse

Keyword(s):

Receptor Antagonist ◽

Gastric Ph ◽

Cyp3a4 Inducer

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Effects of H2-receptor antagonist famodipine on gastric pH and volume of gastric content in patients undergoing CABG with cardiopulmonary bypass

European Journal of Anaesthesiology ◽

10.1097/00003643-200219271-00024 ◽

2002 ◽

Vol 19 (Supplement 27) ◽

pp. 8

Author(s):

N. Trekova ◽

A. Yavorovsky ◽

M. Shmirin ◽

A. Bunatian

Keyword(s):

Cardiopulmonary Bypass ◽

Receptor Antagonist ◽

Gastric Content ◽

Gastric Ph ◽

H2 Receptor Antagonist ◽

H2 Receptor

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Single oral doses of netazepide (YF476), a gastrin receptor antagonist, cause dose-dependent, sustained increases in gastric pH compared with placebo and ranitidine in healthy subjects

Alimentary Pharmacology & Therapeutics ◽

10.1111/j.1365-2036.2012.05143.x ◽

2012 ◽

Vol 36 (2) ◽

pp. 181-189 ◽

Cited By ~ 23

Author(s):

M. Boyce ◽

O. David ◽

K. Darwin ◽

T. Mitchell ◽

A. Johnston ◽

...

Keyword(s):

Receptor Antagonist ◽

Healthy Subjects ◽

Gastric Ph ◽

Gastrin Receptor ◽

Oral Doses ◽

Dose Dependent

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Faculty Opinions recommendation of Single oral doses of netazepide (YF476), a gastrin receptor antagonist, cause dose-dependent, sustained increases in gastric pH compared with placebo and ranitidine in healthy subjects.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.717548133.793003147 ◽

2012 ◽

Author(s):

Ian Beales

Keyword(s):

Receptor Antagonist ◽

Healthy Subjects ◽

Gastric Ph ◽

Gastrin Receptor ◽

Oral Doses ◽

Dose Dependent

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INTERMITTENT INTRAVENOUS PANTOPRAZOLE RAPIDLY ACHIEVES AND MAINTAINS GASTRIC PH≥4 COMPARED WITH CONTINUOUS INFUSION H2-RECEPTOR ANTAGONIST IN INTENSIVE CARE UNIT (ICU) PATIENTS

Critical Care Medicine ◽

10.1097/00003246-200212001-00117 ◽

2002 ◽

Vol 30 (Supplement) ◽

pp. A34 ◽

Cited By ~ 6

Author(s):

John A Morris

Keyword(s):

Intensive Care Unit ◽

Intensive Care ◽

Receptor Antagonist ◽

Continuous Infusion ◽

Gastric Ph ◽

H2 Receptor Antagonist ◽

Icu Patients ◽

H2 Receptor

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The novel histamine H2 receptor antagonist FRG-8813 prevents delay of wound repair induced by hydrogen peroxide in a rabbit gastric epithelial cell system

Journal of Gastroenterology and Hepatology ◽

10.1046/j.1440-1746.1998.01735.x ◽

1998 ◽

Vol 13 (11-s4) ◽

pp. S209-S213

Author(s):

NOBUHIRO SATO ◽

SUMIO WATANABE ◽

XIAN-EN WANG ◽

TARO OSADA ◽

HIROSHI TANAKA ◽

...

Keyword(s):

Hydrogen Peroxide ◽

Epithelial Cell ◽

Receptor Antagonist ◽

Wound Repair ◽

Cell System ◽

The Novel ◽

H2 Receptor Antagonist ◽

Histamine H2 Receptor ◽

H2 Receptor ◽

Histamine H2 Receptor Antagonist

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Colonic effects of TAK-637: A novel NK, receptor antagonist

Gastroenterology ◽

10.1016/s0016-5085(01)81646-2 ◽

2001 ◽

Vol 120 (5) ◽

pp. A331-A331

Author(s):

K VENKOVA ◽

K TYLER ◽

D SUTKOWSKIMARKMANN

Keyword(s):

Receptor Antagonist ◽

Nk Receptor

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Interleukin-1 regulates interleukin-1β/interleukin-1 receptor antagonist mRNA expression in human endometrial stromal cells

Journal of the Society for Gynecologic Investigation ◽

10.1016/s1071-5576(97)86393-9 ◽

1998 ◽

Vol 5 (1) ◽

pp. 116A-116A

Author(s):

H HUANG ◽

Y WEN ◽

J KRUSSEL ◽

H WANG ◽

Y SOONG ◽

...

Keyword(s):

Receptor Antagonist ◽

Mrna Expression ◽

Stromal Cells ◽

Interleukin 1 ◽

Interleukin 1Β ◽

Endometrial Stromal Cells ◽

Interleukin 1 Receptor Antagonist

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Continuous brachial plexus blockade in combination with the NMDA receptor antagonist memantine prevents phantom pain in acute traumatic upper limb amputees

Yearbook of Anesthesiology and Pain Management ◽

10.1016/s1073-5437(08)70995-1 ◽

2008 ◽

Vol 2008 ◽

pp. 265-266

Author(s):

S.E. Abram

Keyword(s):

Nmda Receptor ◽

Brachial Plexus ◽

Receptor Antagonist ◽

Upper Limb ◽

Nmda Receptor Antagonist ◽

Phantom Pain ◽

Brachial Plexus Blockade

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Abstract #1229: Effects on Glucose Lowering of a Cortisol Receptor Antagonist in Cushing Syndrome

Endocrine Practice ◽

10.1016/s1530-891x(20)42458-9 ◽

2015 ◽

Vol 21 ◽

pp. 289

Author(s):

Amy Lee

Keyword(s):

Receptor Antagonist ◽

Cushing Syndrome ◽

Glucose Lowering

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Effects of rolofylline, a new adenosine A1 receptor antagonist, on symptoms, renal function and outcomes in patients with acute heart failure. Results of the PROTECT pilot study

European Journal of Heart Failure Supplements ◽

10.1016/s1567-4215(08)60149-6 ◽

2008 ◽

Vol 7 ◽

pp. 53-54

Author(s):

C OCONNOR ◽

G COTTER ◽

H DITTRICH ◽

B DAVISONWEATHERLEY ◽

M METRA ◽

...

Keyword(s):

Heart Failure ◽

Renal Function ◽

Pilot Study ◽

Receptor Antagonist ◽

Acute Heart Failure ◽

Adenosine A1 Receptor ◽

Adenosine A1 ◽

A1 Receptor

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