A non-calcemic sulfone version of the vitamin D3 analogue seocalcitol (EB 1089): chemical synthesis, biological evaluation and potency enhancement of the anticancer drug adriamycin

G Posner

doi:10.1016/s0968-0896(01)00159-6

A non-calcemic sulfone version of the vitamin D3 analogue seocalcitol (EB 1089): chemical synthesis, biological evaluation and potency enhancement of the anticancer drug adriamycin

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(01)00159-6 ◽

2001 ◽

Vol 9 (9) ◽

pp. 2365-2371 ◽

Cited By ~ 20

Author(s):

G Posner

Keyword(s):

Chemical Synthesis ◽

Anticancer Drug ◽

Vitamin D3 ◽

Biological Evaluation ◽

Eb 1089

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Chemical Synthesis, in vitro Biological Evaluation and Theoretical Investigations of Transition Metal Complexes Derived from 2-(((5-mercapto-1H-pyrrol-2-yl)imino) methyl)6-methoxyphenol

Journal of Molecular Structure ◽

10.1016/j.molstruc.2021.130920 ◽

2021 ◽

pp. 130920

Author(s):

Honnalagere Mariswamy Vinusha ◽

Shiva Prasad Kollur ◽

Muneera Begum ◽

Chandan Shivamallu ◽

Ramith Ramu ◽

...

Keyword(s):

Transition Metal ◽

Chemical Synthesis ◽

Metal Complexes ◽

Transition Metal Complexes ◽

Biological Evaluation ◽

Theoretical Investigations

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Chemical synthesis and preliminary biological evaluation of C-6-O-methyl-1-deoxynojirimycin as a potent α-glucosidase inhibitor

Journal of Carbohydrate Chemistry ◽

10.1080/07328303.2019.1700995 ◽

2019 ◽

Vol 39 (1) ◽

pp. 36-49 ◽

Cited By ~ 1

Author(s):

Lin Wang ◽

Tingting Liang ◽

Zhijie Fang

Keyword(s):

Chemical Synthesis ◽

Biological Evaluation ◽

Glucosidase Inhibitor

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Synthesis and biological evaluation of novel 1-O- and 14-O-derivatives of oridonin as potential anticancer drug candidates

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2008.06.097 ◽

2008 ◽

Vol 18 (16) ◽

pp. 4741-4744 ◽

Cited By ~ 47

Author(s):

Jinyi Xu ◽

JingYi Yang ◽

Qian Ran ◽

Lei Wang ◽

Jie Liu ◽

...

Keyword(s):

Anticancer Drug ◽

Biological Evaluation ◽

Drug Candidates ◽

Synthesis And Biological Evaluation ◽

Derivatives Of

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ChemInform Abstract: Overview of a Rational Approach to Design Type I 17β-Hydroxysteroid Dehydrogenase Inhibitors Without Estrogenic Activity: Chemical Synthesis and Biological Evaluation

ChemInform ◽

10.1002/chin.199904257 ◽

2010 ◽

Vol 30 (4) ◽

pp. no-no

Author(s):

M. R. TREMBLAY ◽

D. POIRIER

Keyword(s):

Chemical Synthesis ◽

Estrogenic Activity ◽

Hydroxysteroid Dehydrogenase ◽

Biological Evaluation ◽

Rational Approach ◽

Type I ◽

Design Type ◽

Synthesis And Biological Evaluation

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Chemical synthesis and biological activity of 3-deoxy-1α-hydroxyvitamin D3 an analog of 1α,25-(OH)2-D3, the active form of vitamin D3

Biochemical and Biophysical Research Communications ◽

10.1016/0006-291x(74)90189-2 ◽

1974 ◽

Vol 60 (1) ◽

pp. 179-185 ◽

Cited By ~ 28

Author(s):

William H. Okamura ◽

Manindra N. Mitra ◽

Richard M. Wing ◽

Anthony W. Norman

Keyword(s):

Biological Activity ◽

Chemical Synthesis ◽

Vitamin D3 ◽

Active Form

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Potentiation of cell killing by fractionated radiation and suppression of proliferative recovery in MCF-7 breast tumor cells by the Vitamin D3 analog EB 1089

The Journal of Steroid Biochemistry and Molecular Biology ◽

10.1016/j.jsbmb.2004.07.011 ◽

2004 ◽

Vol 92 (5) ◽

pp. 365-374 ◽

Cited By ~ 16

Author(s):

Gerald A. DeMasters ◽

Mona S. Gupta ◽

Kara R. Jones ◽

Myles Cabot ◽

Hongtao Wang ◽

...

Keyword(s):

Tumor Cells ◽

Vitamin D3 ◽

Breast Tumor ◽

Cell Killing ◽

Breast Tumor Cells ◽

Eb 1089 ◽

Fractionated Radiation ◽

Mcf 7

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Chemical Synthesis ofEscherichia ColiSThAnalogues by Regioselective Disulfide Bond Formation: Biological Evaluation of an111In-DOTA−Phe19-SThAnalogue for Specific Targeting of Human Colon Cancers

Bioconjugate Chemistry ◽

10.1021/bc010062u ◽

2002 ◽

Vol 13 (2) ◽

pp. 224-231 ◽

Cited By ~ 20

Author(s):

Hariprasad Gali ◽

Gary L. Sieckman ◽

Timothy J. Hoffman ◽

Nellie K. Owen ◽

Dana G. Mazuru ◽

...

Keyword(s):

Chemical Synthesis ◽

Disulfide Bond ◽

Bond Formation ◽

Human Colon ◽

Biological Evaluation ◽

Disulfide Bond Formation ◽

Specific Targeting ◽

Colon Cancers

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Molecular docking, structure–activity relationship and biological evaluation of the anticancer drug monastrol as a pteridine reductase inhibitor in a clinical isolate of Leishmania donovani

Journal of Antimicrobial Chemotherapy ◽

10.1093/jac/dkq189 ◽

2010 ◽

Vol 65 (8) ◽

pp. 1742-1748 ◽

Cited By ~ 24

Author(s):

Jaspreet Kaur ◽

Shyam Sundar ◽

Neeloo Singh

Keyword(s):

Molecular Docking ◽

Clinical Isolate ◽

Anticancer Drug ◽

Reductase Inhibitor ◽

Leishmania Donovani ◽

Structure Activity Relationship ◽

Biological Evaluation ◽

Activity Relationship ◽

Structure Activity

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Chemical synthesis and biological evaluation of a NAD(P)H:quinone oxidoreductase-1 targeted tripartite quinone drug delivery system

Molecular Cancer Therapeutics ◽

10.1158/1535-7163.mct-07-0519 ◽

2007 ◽

Vol 6 (12) ◽

pp. 3122-3130 ◽

Cited By ~ 25

Author(s):

M. Volpato ◽

N. Abou-Zeid ◽

R. W. Tanner ◽

L. T. Glassbrook ◽

J. Taylor ◽

...

Keyword(s):

Drug Delivery ◽

Chemical Synthesis ◽

Drug Delivery System ◽

Delivery System ◽

Biological Evaluation ◽

Synthesis And Biological Evaluation

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Chemical Synthesis and Biological Evaluation of Second-Generation Palmerolide A Analogues

European Journal of Organic Chemistry ◽

10.1002/ejoc.201001562 ◽

2010 ◽

Vol 2011 (3) ◽

pp. 463-468 ◽

Cited By ~ 14

Author(s):

Vengala Rao Ravu ◽

Gulice Y. C. Leung ◽

Chek Shik Lim ◽

Sin Yee Ng ◽

Rong Ji Sum ◽

...

Keyword(s):

Chemical Synthesis ◽

Second Generation ◽

Biological Evaluation ◽

Palmerolide A ◽

Synthesis And Biological Evaluation

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