Synthesis of constrained analogues of tryptophan
2015 ◽
Vol 11
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pp. 1997-2006
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A Lewis acid-catalysed diastereoselective [4 + 2] cycloaddition of vinylindoles and methyl 2-acetamidoacrylate, leading to methyl 3-acetamido-1,2,3,4-tetrahydrocarbazole-3-carboxylate derivatives, is described. Treatment of the obtained cycloadducts under hydrolytic conditions results in the preparation of a small library of compounds bearing the free amino acid function at C-3 and pertaining to the class of constrained tryptophan analogues.
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1962 ◽
2013 ◽
Vol 42
(1)
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pp. 96-101
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2020 ◽
Vol 23
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Keyword(s):
2020 ◽
Vol 22
(9)
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pp. 657-662
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1971 ◽
Vol 11
(1)
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pp. 112-114
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2006 ◽
Vol 12
(3)
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pp. 199-205
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